Aprocitentan
Products
Description
Aprocitentan (ACT-132577) is a pharmacologically active metabolite of Macitentan. Aprocitentan is an orally active dual antagonist of ETA/ETB with IC50 values of 3.4 nM and 987 nM, and pA2 values of 6.7 and 5.5, respectively.
Specifications
| Manufacturer Cat# | E4771 |
|---|---|
| Target | Endothelin Receptor |